Inhibitors | Comment | Organism | Structure |
---|---|---|---|
convallatoxin | - |
Homo sapiens | |
digitoxigenin | - |
Homo sapiens | |
digitoxin | - |
Homo sapiens | |
digoxin | - |
Homo sapiens | |
additional information | cardiac glycosides can dramatically suppress the transcription of KLKs | Homo sapiens | |
Ouabain | - |
Homo sapiens | |
peruvoside | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
MDA-MB-468 cell | - |
Homo sapiens | - |
Synonyms | Comment | Organism |
---|---|---|
KLK5 | - |
Homo sapiens |
KLK6 | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.000006 | - |
KLK6 | Homo sapiens | peruvoside | |
0.000008 | - |
KLK5 | Homo sapiens | peruvoside | |
0.000042 | - |
KLK5 | Homo sapiens | digitoxin | |
0.00005 | - |
KLK6 | Homo sapiens | digitoxin | |
0.000065 | - |
KLK6 | Homo sapiens | Ouabain | |
0.00009 | - |
KLK5 | Homo sapiens | digoxin | |
0.0001 | - |
KLK6 | Homo sapiens | digoxin | |
0.00012 | - |
KLK5 | Homo sapiens | Ouabain | |
0.00013 | - |
KLK6 | Homo sapiens | convallatoxin | |
0.00015 | - |
KLK5 | Homo sapiens | convallatoxin | |
0.00021 | - |
KLK5 | Homo sapiens | digitoxigenin | |
0.00038 | - |
KLK6 | Homo sapiens | digitoxigenin |